Synthesis of Benzofuran Derivatives through Cascade Radical Cyclization/Intermolecular Coupling of 2-AzaallylsBy: Deng, GG (Deng, Guogang) [1] ; Li, MY (Li, Minyan)[2] ; Yu, KL (Yu, Kaili)[1] ; Liu, CX (Liu, Chunxiang)[1] ; Liu, ZF (Liu, Zhengfen)[1] ; Duan, SZ (Duan, Shengzu)[1] ; Chen, W (Chen, Wen)[1] ; Yang, XD (Yang, Xiaodong)[1] ; Zhang, HB (Zhang, Hongbin)[1] ; Walsh, PJ (Walsh, Patri...
Palladium-Catalyzed Alkenylation of Azaarylmethylamines with Vinyl HalidesBy: Duan, Shengzu; Li, Minyan; Ma, Xueqiong; Chen, Wen; Li, Liang; Zhang, Hongbin; Yang, Xiaodong; Walsh, Patrick J. ADVANCED SYNTHESIS & CATALYSISVolume:360Issue:24Pages:4837-4842DOI:10.1002/adsc.201801045Published:DEC 21 2018Document Type:ArticleADVANCED SYNTHESIS & CATALYSIS Impact Factor5.1235.02920175 yearJCR® ...
B591,a novel specific pan-PI3K inhibitor,preferentially targets cancer stem cellsBy: Zhou, Hongyu;Yu, Chunlei;Kong, Lingmei;Xu, Xiaoliang;Yan, Juming;Li, Yingchao;An, Tao;Gong, Liang;Gong, Yaxiao;Zhu, Huifang...MoreOncogeneDOI:10.1038/s41388-018-0674-5Published:2019-Jan-11(Epub 2019 Jan 11)Document Type: Journal ArticleAbstractCancer stem cells (CSCs) have been implicated in metastasis, relapse...
Cascade Reaction of Morita–Baylis–Hillman Acetates with 1,1-Enediamines or Heterocyclic Ketene Aminals: Synthesis of Highly Functionalized 2-AminopyrrolesJin Liu , Qi Li, Zheng-Mao Cao, Yi Jin , Jun Lin* , and Sheng-Jiao Yan* Key Laboratory of Medicinal Chemistry for Natural Resource (Yunnan University), Ministry of Education, School of Chemical Science and Technology , Yunna...
Chemical Space and Biological Target Network of Anti-Inflammatory Natural ProductsRuihan Zhang, Jing Lin, Yan Zou, Xing-Jie Zhang, and Wei-Lie Xiao* Key Laboratory of Medicinal Chemistry for Natural Resources, Ministry of Education and Yunnan Province, School of Chemical Science and Technology, Yunnan University, 2Rd. Cuihubei, Kunming 650091 , ChinaJournal of Chemical Information and Mo...
Highly Selective Synthesis of 2-Amino-4,6-diarylpyridine Derivatives by the Cascade Reaction of 1,1-Enediamines with α,β-Unsaturated KetonesQin Luo†, Rong Huang†, Qiang Xiao, Yuan Yao, Jun Lin* , and Sheng-Jiao Yan* Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education, School of Chemical Science and Technology, Yunnan University , Kunming 650091...
Three-Component Cascade Reaction of 1,1-Enediamines, N,N‑Dimethylformamide Dimethyl Acetal, and 1,3-Dicarbonyl Compounds: Selective Synthesis of Diverse 2‑Aminopyridine DerivativesBY: Quan-Xing Zi, Sheng-Jiao Yan,* Chang-Long Yang, Kun Li, and Jun Lin*Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education and Yunnan Province, School of Chemical Science and Technolog...
Transition-metal-free a-arylation of oxindoles via visible-light-promoted electron transferBY: Kangjiang Liang, Na Li, Yang Zhang, Tao Li and Chengfeng Xia*Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education and Yunnan Province, School of Chemical Science and Technology, Yunnan University , Kunming 650091 , P. R. China Chemical ScienceDOI: 10.1039/c8...
Enantioselective Epoxypyrrolidines via a Tandem Cycloaddition/Autoxidation in Air and Mechanistic StudiesBY: Kaixiu Luo, Yongqiang Zhao, Jiawei Zhang, Jia He, Rong Huang, Shengjiao Yan*, Jun Lin*, and Yi Jin*Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education and Yunnan Province, School of Chemical Science and Technology, Yunnan University , Kunming 65...
Total synthesis of (−)-vindolineBy: Wen Chen, Hongchang Tian, Wenyun Tan, Xiaotong Liu, Xiaodong Yang, Hongbin ZhangKey Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education and Yunnan Province, School of Chemical Science and Technology, Yunnan University, Kunming, Yunnan, 650091, People's Republic of ChinaTetrahedronAvailable online 28 November 2018 AbstractIn this fu...